99.4% Purity
In Stock
Tirzepatide (15mg)
- Tirzepatide (LY3298176) is a first-in-class 39-amino acid dual GIP/GLP-1 receptor agonist ("twincretin") with imbalanced agonism favoring GIPR over GLP-1R
- Features Aib residues at positions 2 and 13 (DPP-4 resistance), C20 fatty diacid at Lys20 (albumin binding, ~5-day half-life), and biased GLP-1R signaling favoring cAMP over beta-arrestin recruitment
- FDA-approved as Mounjaro (T2D, May 2022) and Zepbound (obesity, Nov 2023)
$129.00